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11793

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8607 (73.0%)
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6418 (54.4%)
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11793 (100.0%)

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Halaman 100 / 236
Farglitazar DB19311
small molecule | CAS: 274687-78-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
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Faricimab Approved DB15303
biotech | CAS: 1607793-29-2

Retinal vascular diseases (RVDs) such as diabetic macular edema (DME), age-related macular degeneration (AMD), and retinal vein occlusion (RVO) are typically caused by retinal ischemia and subsequent neovascularization (NV).[A225985, A225990, A225995] Vascula…

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +15
Target Protein:
Vascular endothelial growth factor A, long formAngiopoietin-2
Waktu ParuhFaricimab has an es…
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Farletuzumab DB05595
biotech | CAS: 896723-44-7

Farletuzumab (MORAb-003) is a fully humanized monoclonal antibody against the folate receptor alpha, for the potential treatment of epithelial ovarian cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Folate receptor alpha
Waktu Paruh-
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biotech | CAS: 2407465-18-1

Farletuzumab ecteribulin is under investigation in clinical trial NCT04300556 (A Study to Evaluate the Safety, Tolerability, and Efficacy of Morab-202 (Herein Referred to as Farletuzumab Ecteribulin), a Folate Receptor Alpha (Fr?)-targeting Antibody-drug Conj…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
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Farnesol DB02509
small molecule | CAS: 4602-84-0

A colorless liquid extracted from oils of plants such as citronella, neroli, cyclamen, and tuberose. It is an intermediate step in the biological synthesis of cholesterol from mevalonic acid in vertebrates. It has a delicate odor and is used in perfumery. (Fr…

Kategori:
AlcoholsFatty AlcoholsLipids +2
Target Protein:
Amine oxidase [flavin-containing] BBile acid receptor
Waktu Paruh-
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Genetik -
small molecule | CAS: 13058-04-3

Deskripsi belum tersedia.

Kategori:
OrganophosphatesOrganophosphorus CompoundsPotential QTc-Prolonging Agents +2
Target Protein:
Squalene synthaseProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaProtein farnesyltransferase subunit beta +9
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
OrganophosphatesOrganophosphorus CompoundsPotential QTc-Prolonging Agents +2
Target Protein:
Geranylgeranyl pyrophosphate synthaseMevalonate kinaseDehydrosqualene synthase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Faropenem DB12190
small molecule | CAS: 106560-14-9

Faropenem has been used in trials studying the treatment of Tuberculosis, Pulmonary Tuberculosis, and Community Acquired Pneumonia.

Kategori:
AmidesAntibacterials for Systemic UseAntiinfectives for Systemic Use +3
Target Protein:
Dihydropteroate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 141702-36-5

Faropenem medoxomil is an ester prodrug derivative of the beta-lactam antibiotic [faropenem]. The prodrug form of faropenem offers dramatically improved oral bioavailability and leads to higher systemic concentrations of the drug. Faropenem medoxomil is a bro…

Kategori:
AmidesHeterocyclic Compounds, Fused-RingLactams +1
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 2BPeptidoglycan D,D-transpeptidase FtsI
Waktu Paruh-
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Farudodstat DB16049
small molecule | CAS: 1035688-66-4

Farudodstat (ASLAN003) is under investigation in clinical trial NCT03451084 (A Dose Optimisation Study of ASLAN003 in Acute Myeloid Leukemia).

Kategori:
AminesEnzyme InhibitorsPyridines
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Fasentin DB16759
small molecule | CAS: 392721-37-8

Deskripsi belum tersedia.

Kategori:
AmidesAminesAniline Compounds
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Fasinumab DB12157
biotech | CAS: 1190239-42-9

Fasinumab is a human IgG1k monoclonal antibody targeted against nerve growth factor (NGF). It is currently under investigation for the treatment osteoarthritic pain[A241045] and has demonstrated significantly greater pain relief and functional improvement as …

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +11
Target Protein:
Beta-nerve growth factor
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Fasitibant DB15646
small molecule | CAS: 869939-83-3

Fasitibant is under investigation in clinical trial NCT02205814 (Fasitibant Intra-articular Injection in Patients With Symptomatic Osteoarthritis of the Knee).

Kategori:
AmidesAmino AcidsAmino Acids, Basic +9
Target Protein:
B2 bradykinin receptor
Waktu Paruh-
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Fasoracetam DB16163
small molecule | CAS: 110958-19-5

Fasoracetam is under investigation in clinical trial NCT03609619 (PART B: Efficacy and Safety of AEVI-001 in Children and Adolescents With ADHD and Without Mglur Mutations).

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +2
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Fasudil DB08162
small molecule | CAS: 103745-39-7

Fasudil has been investigated in Carotid Stenosis.

Kategori:
Antiarrhythmic agentsCalcium Channel BlockersCalcium-Regulating Hormones and Agents +12
Target Protein:
Rho-associated protein kinase 1cAMP-dependent protein kinase inhibitor alphacAMP-dependent protein kinase catalytic subunit alpha +1
Waktu Paruh-
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Genetik -
FAV-201 DB06130
biotech

FAV-201 is a patient-specific immunotherapy for the treatment of T-cell lymphoma.

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Favezelimab DB16729
biotech | CAS: 2231068-83-8

Favezelimab is under investigation in clinical trial NCT04626479 (Substudy 03A: A Study of Immune and Targeted Combination Therapies in Participants With First Line (1L) Renal Cell Carcinoma (MK-3475-03A)).

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Favipiravir Approved DB12466
small molecule | CAS: 259793-96-9

Discovered by Toyama Chemical Co., Ltd. in Japan, favipiravir is a modified pyrazine analog that was initially approved for therapeutic use in resistant cases of influenza.[A191688,A191721] The antiviral targets RNA-dependent RNA polymerase (RdRp) enzymes, wh…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +11
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'RNA-directed RNA polymerase catalytic subunit
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe recommended ora…
Genetik -
small molecule | CAS: 49564-56-9

Deskripsi belum tersedia.

Kategori:
Central Nervous System DepressantsMuscle RelaxantsMuscle Relaxants, Peripherally Acting Agents +2
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Fazirsiran DB17891
biotech | CAS: 2175009-08-0

Deskripsi belum tersedia.

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Fazpilodemab DB18924
biotech | CAS: 2517935-02-1

Fazpilodemab is under investigation in clinical trial NCT04171765 (A Study to Evaluate the Efficacy, Safety, and Pharmacokinetics of BFKB8488A Compared With Placebo in Participants With Non-alcoholic Steatohepatitis).

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FB-101 DB17956
small molecule

FB-101 is a c-Abl inhibitor. Developed by 1st Biotherapeutics, it is being investigated for the treatment of neurological disorders, such as Parkinson's Disease and amyotrophic lateral sclerosis (ALS).[L47102]

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fb-PMT DB17394
small molecule

Deskripsi belum tersedia.

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FDL169 DB16878
small molecule | CAS: 1628416-28-3

Deskripsi belum tersedia.

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Febantel DB11409
small molecule | CAS: 58306-30-2

Deskripsi belum tersedia.

Kategori:
AmidinesAnthelminticsAnti-Infective Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Febarbamate DB13303
small molecule | CAS: 13246-02-1

Deskripsi belum tersedia.

Kategori:
Carbamic Acid EstersCentral Nervous System DepressantsMuscle Relaxants +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Febuxostat Approved DB04854
small molecule | CAS: 144060-53-7

Febuxostat is a non-purine xanthine oxidase (XO) inhibitor.[A39743] In early 2008, febuxostat was granted marketing authorization by the European Commission for the treatment of chronic hyperuricemia and gout.[A230548] In the following year, the FDA for appro…

Kategori:
Antigout PreparationsAntirheumatic AgentsBCRP/ABCG2 Inhibitors +15
Target Protein:
Xanthine dehydrogenase/oxidase
Waktu ParuhThe apparent mean t…
Vol. DistribusiThe apparent steady…
KlirensFollowing oral admi…
Genetik -
Fecal microbiota Approved DB17743
biotech

Fecal microbiota, given either as a rectal transplant or in an oral formulation of live spores, is an FDA-approved option to prevent the recurrence of _Clostridioides difficile_ infection (CDI) in patients given an antibacterial treatment for recurrent CDI.[A…

Kategori:
Miscellaneous Therapeutic Agents
Waktu ParuhNot available.
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Fedovapagon DB11734
small molecule | CAS: 347887-36-9

Fedovapagon has been used in trials studying the treatment of Nocturia.

Target Protein:
Vasopressin V2 receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Fedratinib Approved DB12500
small molecule | CAS: 936091-26-8

Fedratinib, also known as SAR302503 and TG101348, is a tyrosine kinase inhibitor used to treat intermediate-2 and high risk primary and secondary myelofibrosis.[A183176,L8090] It is an anilinopyrimidine derivative.[A183188] Fedratinib was granted FDA appro…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +25
Target Protein:
Tyrosine-protein kinase JAK2Receptor-type tyrosine-protein kinase FLT3Tyrosine-protein kinase JAK1
Waktu ParuhThe half life of fe…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of fe…
Genetik -
Feladilimab DB16415
biotech

Feladilimab is under investigation in clinical trial NCT04128696 (Study of GSK3359609 and Pembrolizumab in Programmed Death Receptor 1-ligand 1 Positive Recurrent or Metastatic Head and Neck Squamous Cell Carcinoma).

Waktu Paruh-
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Felcisetrag DB12725
small molecule | CAS: 916075-84-8

Felcisetrag (TD-8954) has been used in trials studying the treatment of Enteral Feeding Intolerance and Gastrointestinal Motility Disorder.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
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Genetik -
Felodipine Approved DB01023
small molecule | CAS: 72509-76-3

Felodipine is a long-acting 1,4-dihydropyridine calcium channel blocker (CCB)b. It acts primarily on vascular smooth muscle cells by stabilizing voltage-gated L-type calcium channels in their inactive conformation. By inhibiting the influx of calcium in smoot…

Kategori:
ACE Inhibitors and Calcium Channel BlockersAgents causing hyperkalemiaAntiarrhythmic agents +31
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent L-type calcium channel subunit beta-2 +10
Waktu Paruh17.5-31.5 hours in …
Vol. Distribusi* 10 L/kg
Klirens* 0.8 L/min [Young …
Genetik -
Felypressin DB00093
biotech | CAS: 56-59-7

A synthetic nonapeptide comprising cysteinyl, phenylalanyl, phenylalanyl, glutaminyl, asparaginyl, cysteinyl, prolyl, lysyl, and glycinamide residues in sequence, with a disulfide bridge joining the two cysteine residues. Its antidiuretic effects are less tha…

Kategori:
Amino Acids, Peptides, and ProteinsCardiovascular AgentsHormones +12
Target Protein:
Vasopressin V1a receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Felzartamab DB16375
biotech | CAS: 2197112-39-1

Felzartamab is under investigation in clinical trial NCT04145440 (Trial to Assess Safety and Efficacy of MOR202 in Anti-pla2r + Membranous Nephropathy (Amn)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
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Fenamole DB12506
small molecule | CAS: 5467-78-7

Fenamole has been investigated for the supportive care of Side Effects and Dental Plaque.

Waktu Paruh-
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Fenbendazole DB11410
small molecule | CAS: 43210-67-9

Fenbendazole is a benzimidazole that presents a wide spectrum anthelmintic effect. It is used against a number of gastrointestinal parasites including giardia, roundworms, hookworms, whipworms, the Taenia genus of tapeworms, pinworms, aelurostrongylus, parago…

Kategori:
Acids, AcyclicAnthelminticsAnti-Infective Agents +7
Waktu Paruh-
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Genetik -
Fenbufen Approved DB08981
small molecule | CAS: 36330-85-5

Fenbufen is a non-steroidal anti-inflammatory drug used primarily to treat inflammation in osteoarthritis, ankylosing spondylitis, and tendinitis. It can also be used to relieve backaches, sprains, and fractures. Fenbufen is available as a capsule or tablet s…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +15
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh-
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Fencamfamin DB01463
small molecule | CAS: 1209-98-9

Fencamfamin (Glucoenergan, Reactivan) is a stimulant which was developed in the 1960s as an appetite suppressant, but was later withdrawn for this application due to problems with dependence and abuse. It is around half the potency of [dexamphetamine], and is…

Kategori:
Bridged-Ring CompoundsCentral Nervous System AgentsCentral Nervous System Depressants +7
Target Protein:
Sodium-dependent dopamine transporterD(2) dopamine receptor
Waktu Paruh-
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Fenebrutinib DB14785
small molecule | CAS: 1434048-34-6

Fenebrutinib is under investigation in clinical trial NCT03174041 (A Drug-Drug Interaction Study Between GDC-0853 and Midazolam, Itraconazole, Rosuvastatin, and Simvastatin).

Kategori:
Pyridines
Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
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Fenethylline DB01482
small molecule | CAS: 3736-08-1

Deskripsi belum tersedia.

Kategori:
AlkaloidsAminesCentral Nervous System Agents +13
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Fenfluramine Approved DB00574
small molecule | CAS: 458-24-2

Dravet syndrome is a pediatric encephalopathy that typically manifests within the first year of life following exposure to elevated temperatures. It is characterized by recurrent pharmacoresistant seizures, which increase in frequency and severity with diseas…

Kategori:
Alimentary Tract and MetabolismAminesAnticonvulsants +27
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 2C +4
Waktu ParuhFenfluramine has an…
Vol. DistribusiFenfluramine has an…
KlirensFenfluramine has a …
Genetik -
Fennel Approved DB15615
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Fenobam DB12931
small molecule | CAS: 57653-26-6

Fenobam is under investigation in clinical trial NCT00637221 (Open Label Study Investigating Safety and Efficacy of Fenobam anhydrous 50 mg - 150 mg on Prepulse Inhibition Tests and Continuous Performance Tasks, Adults With Fragile X Syndrome).

Target Protein:
Metabotropic glutamate receptor 5
Waktu Paruh-
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Genetik -
Fenofibrate Approved DB01039
small molecule | CAS: 49562-28-9

Fenofibrate is a fibric acid derivative like [clofibrate] and [gemfibrozil].[A185954] Fenofibrate is used to treat primary hypercholesterolemia, mixed dyslipidemia, severe hypertriglyceridemia.[L8588,L8591] Fenofibrate was granted FDA approval on 31 Decemb…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityBenzene Derivatives +39
Target Protein:
Peroxisome proliferator-activated receptor alphaNuclear receptor subfamily 1 group I member 2Matrix metalloproteinase-25
Waktu ParuhFenofibric acid, th…
Vol. DistribusiThe volume of distr…
KlirensThe oral clearance …
Genetik -
Fenofibric acid Approved DB13873
small molecule | CAS: 42017-89-0

Fenofibric acid is a lipid-lowering agent that is used in severe hypertriglyceridemia, primary hyperlipidemia, and mixed dyslipidemia. It works to decrease elevated low-density lipoprotein cholesterol, total cholesterol, triglycerides, apolipoprotein B, while…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityAnticholesteremic Agents +17
Target Protein:
Peroxisome proliferator-activated receptor alphaFatty acid-binding protein, liverMatrix metalloproteinase-25 +3
Waktu ParuhFollowing once dail…
Vol. DistribusiThe volume of distr…
KlirensIn five elderly vol…
Genetik -
Fenoldopam Approved DB00800
small molecule | CAS: 67227-56-9

A dopamine D1 receptor agonist that is used as an antihypertensive agent. It lowers blood pressure through arteriolar vasodilation.

Kategori:
Adrenergic and Dopaminergic AgentsAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +12
Target Protein:
D(1B) dopamine receptorD(1A) dopamine receptorAlpha-1B adrenergic receptor +5
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Fenoprofen Approved DB00573
small molecule | CAS: 29679-58-1

An anti-inflammatory analgesic and antipyretic highly bound to plasma proteins. It is pharmacologically similar to aspirin, but causes less gastrointestinal bleeding.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +18
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1Peroxisome proliferator-activated receptor alpha +1
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
Genetik -
Fenoverine DB13042
small molecule | CAS: 37561-27-6

Fenoverine has been used in trials studying the treatment of Irritable Bowel Syndrome.

Kategori:
Alimentary Tract and MetabolismAutonomic AgentsDrugs for Functional Gastrointestinal Disorders +4
Waktu Paruh-
Vol. Distribusi-
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small molecule | CAS: 66441-23-4

Fenoxaprop-ethyl (organic nitrate combined with L-arginine), is an oral proprietary nitrate therapeutic shown to induce coronary vasodilation while overcoming the significant problem of drug tolerance. Fenoxaprop-ethyl has been investigated to treat chronic a…

Kategori:
Acids, AcyclicAgrochemicalsCompounds used in a research, industrial, or household setting +6
Target Protein:
Nitric oxide synthase 3Nitric oxide synthase, inducible
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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