Hasil Filter

3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (3253)

Halaman 10 / 66
Balsam of Peru DB11482
small molecule | CAS: 8007-00-9

Balsam of Peru is a resin that comes from the tree Myroxylon balsamum pereirae. It is constituted by a mixture of substances from which the major components are benzyl cinnamate and [DB00676]. Balsam of Peru has also presented several allergens such as cinnam…

Kategori:
Biological ProductsBiopolymersCell-mediated Immunity +8
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Balugrastim DB12699
biotech | CAS: 527698-09-5

Balugrastim has been used in trials studying the treatment of Solid Tumors.

Kategori:
Adjuvants, ImmunologicAlbuminsAmino Acids, Peptides, and Proteins +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bamosiran DB12256
biotech | CAS: 1337968-84-9

Bamosiran has been used in trials studying the treatment of Glaucoma, Ocular Hypertension, and Open Angle Glaucoma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bardoxolone DB12651
small molecule | CAS: 218600-44-3

Bardoxolone has been used in trials studying the treatment of LYMPHOMA and Solid Tumors. It is a synthetic triterpenoid and a highly potent activator of redox-sensitive signaling pathways that induce programmed cell death (apoptosis) in cancer cells that are …

Kategori:
Pentacyclic TriterpenesSapogeninsTerpenes +1
Target Protein:
Nitric oxide synthase, inducibleCaspase-8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Barium DB12481
small molecule | CAS: 7440-39-3

Barium is under investigation for the diagnostic of Known or Suspected Abdominal Disease.

Kategori:
ElementsMetalsMetals, Alkaline Earth +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Barusiban DB12292
small molecule | CAS: 285571-64-4

Barusiban has been used in trials studying the treatment of Infertility and In Vitro Fertilisation (IVF) Treatment.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesReceptors, Oxytocin, antagonists & inhibitors
Target Protein:
Oxytocin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Basifungin DB14058
small molecule | CAS: 127785-64-2

Basifungin, also known as _aureuobacidin A_, is a phosphorylceramide synthase inhibitor [L2960], [A33381].

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +3
Target Protein:
Inositol phosphorylceramide synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Batefenterol DB12526
small molecule | CAS: 743461-65-6

Batefenterol has been used in trials studying the treatment of Pulmonary Disease, Chronic Obstructive.

Kategori:
Acids, AcyclicAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +5
Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bavdegalutamide DB19032
small molecule | CAS: 2222112-77-6

Bavdegalutamide is under investigation in clinical trial NCT03888612 (Trial of ARV-110 in Patients With Metastatic Castration Resistant Prostate Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bavisant DB12299
small molecule | CAS: 929622-08-2

Bavisant has been used in trials studying the basic science and treatment of Alcoholism, Pharmacokinetics, Drug Interactions, Attention Deficit Hyperactivity Disorder, and Attention Deficit Disorders With Hyperactivity.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Histamine H3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BB 21217 DB17373
biotech

BB 21217 is an anti-BCMA CAR T cell therapy that uses the same CAR molecule as [idecabtagene vicleucel] (bb2121), but adds the PI3K inhibitor bb007 during ex vivo culture to enrich the drug product (DP) for memory-like T cells.[L44291]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BB-301 DB17011
biotech

BB-301 is a modified AAV serotype 9 (AAV9) capsid expressing a unique, single bifunctional construct promoting co-expression of both codon-optimized Poly-A Binding Protein Nuclear-1 (PABPN1) and two small inhibitory RNAs (siRNAs) against mutant PABPN1.[A26011…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBP-812 DB16983
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BC9KBY85WY DB17820
small molecule | CAS: 1259013-14-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BCG vaccine Approved DB12768
biotech

BCG vaccine has been investigated for the treatment of Neoplasms, Bladder Cancer, Neoplasms by Site, Urologic Diseases, and Urologic Neoplasms, among others.

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsBacterial Vaccines +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Beclabuvir DB12225
small molecule | CAS: 958002-33-0

Beclabuvir has been used in trials studying the treatment of Hepatitis C, Chronic.

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +3
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bedaquiline Approved DB08903
small molecule | CAS: 843663-66-1

Bedaquiline is a bactericidal antimycobacterial drug belonging to the class of diarylquinoline. The quinolinic central heterocyclic nucleus with alcohol and amine side chains is responsible for bedaquiline-mediated antimycobacterial activity.[A261866] Althoug…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiinfectives for Systemic Use +10
Target Protein:
ATP synthase subunit c
Waktu ParuhThe mean terminal e…
Vol. DistribusiThe volume of distr…
KlirensBedaquiline has a l…
Genetik -
Bee pollen DB16612
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Beeswax Approved DB11600
biotech | CAS: 8012-89-3

The wax obtained from the honeycomb of the bee. It consists primarily of myricyl palmitate, cerotic acid esters and some high-carbon paraffins. Beeswax is used as a stiffening agent in ointments and creams, and enables water to be incorporated to produce wate…

Kategori:
BeesLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Befiradol DB19033
small molecule | CAS: 208110-64-9

Befiradol is under investigation in clinical trial NCT05148884 (Study to Assess the Safety, Tolerability and Preliminary Efficacy of NLX-112 Versus Placebo in L-dopa-induced Dyskinesia).

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsNeurotransmitter Agents +3
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Begacestat DB12263
small molecule | CAS: 769169-27-9

Begacestat has been used in trials studying the treatment and basic science of Alzheimer Disease.

Kategori:
AmidesAmyloid Precursor Protein SecretasesEnzyme Inhibitors +3
Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Beinaglutide DB15072
biotech | CAS: 123475-27-4

Beinaglutide is under investigation in clinical trial NCT03829891 (Study for Beinaglutide Versus Glargine Therapy in Glycemic Variability of Type 2 Diabetes Mellitus).

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Belapectin DB15125
small molecule | CAS: 1980787-47-0

Belapectin is under investigation in clinical trial NCT02575404 (GR-MD-02 Plus Pembrolizumab in Melanoma, Non-small Cell Lung Cancer, and Squamous Cell Head and Neck Cancer Patients).

Kategori:
Biological ProductsBiopolymersCarbohydrates +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Beloranib DB12671
small molecule | CAS: 251111-30-5

Beloranib has been used in trials studying the treatment of Obesity, Over-weight, Type 2 Diabetes, Craniopharyngioma, and Hypothalamic Injury, among others.

Kategori:
Acids, CarbocyclicAngiogenesis InhibitorsAngiogenesis Modulating Agents +7
Target Protein:
Methionine aminopeptidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Belotecan DB12459
small molecule | CAS: 256411-32-2

Belotecan has been investigated for the treatment of Epithelial Ovarian Cancer.

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +4
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Belrestotug DB19066
biotech | CAS: 2574438-65-4

Belrestotug is under investigation in clinical trial NCT05565378 (A Platform Study of Novel Immunotherapy Combinations in Participants With Previously Untreated, Advanced/metastatic Non-small-cell Lung Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Belumosudil Approved DB16703
small molecule | CAS: 911417-87-3

Belumosudil is used in the treatment of chronic graft-versus-host disease (GVHD) and has been investigated for the treatment of pulmonary arterial hypertension.[A236634] It is an inhibitor of rho-associated coiled-coil-containing protein kinases (ROCK), with …

Kategori:
AcetatesAcids, AcyclicAmides +25
Target Protein:
Rho-associated protein kinase 2Rho-associated protein kinase 1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiFollowing a single …
KlirensThe mean clearance …
Genetik -
Bemcentinib DB12411
small molecule | CAS: 1037624-75-1

Bemcentinib has been investigated for the treatment of Non-Small Cell Lung Cancer.

Target Protein:
Spike glycoproteinTyrosine-protein kinase receptor UFO
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bemotrizinol Approved DB11206
small molecule | CAS: 187393-00-6

Bemotrizinol, or bis-ethylhexyloxyphenol methoxyphenyl triazine, is an organic UV filter found in over-the-counter sunscreen products. It primarily absorbs UV-A rays. Compared to older broad-spectrum chemical agents, bemotrizinol is more more fat soluble (oil…

Kategori:
Benzene DerivativesSunscreen Agents
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Bempedoic acid Approved DB11936
small molecule | CAS: 738606-46-7

High levels of LDL cholesterol (LDL-C) are a major risk factor for cardiovascular events. Caused by genetic mutations or lifestyle factors, hypercholesterolemia can significantly reduce quality of life and increase the risk of mortality from cardiovascular di…

Kategori:
Acids, AcyclicAdenosine Triphosphate-Citrate Lyase InhibitorAdenosine Triphosphate-Citrate Lyase Inhibitors +11
Target Protein:
ATP-citrate synthase
Waktu ParuhThe half-life of be…
Vol. DistribusiThe apparent volume…
KlirensThe clearance (CL/F…
Genetik -
biotech | CAS: 1939126-74-5

Bempegaldesleukin is under investigation in clinical trial NCT03729245 (A Study of NKTR-214 in Combination With Nivolumab Compared With the Investigator's Choice of a Tyrosine Kinase Inhibitor (TKI) Therapy (Either Sunitinib or Cabozantinib Monotherapy) for A…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benapenem DB18883
small molecule | CAS: 1312953-83-5

Benapenem is under investigation in clinical trial NCT04505683 (A Study to Assess Efficacy and Safety Intravenous Benapenem in Patients With Complicated Urinary Tract Infection (Cuti) or Acute Pyelonephritis (AP)).

Kategori:
Amidesbeta-LactamsHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benazeprilat DB14125
small molecule | CAS: 86541-78-8

Deskripsi belum tersedia.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benoxaprofen Approved DB04812
small molecule | CAS: 51234-28-7

The use of benoxaprofen, formerly marketed as Oraflex tablets, was associated with fatal cholestatic jaundice among other serious adverse reactions. The holder of the approved application voluntarily withdrew Oraflex tablets from the market on August 5, 1982.

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +18
Target Protein:
Acetyl-CoA acetyltransferase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benperidol Approved DB12867
small molecule | CAS: 2062-84-2

Benperidol has been used in trials studying the treatment of Dementia, Depression, Schizophrenia, Anxiety Disorders, and Psychosomatic Disorders, among others.

Kategori:
Antipsychotic AgentsButyrophenone DerivativesButyrophenones +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benralizumab Approved DB12023
biotech | CAS: 1044511-01-4

Benralizumab is a humanized recombinant monoclonal antibody of the isotype IgG1k immunoglobulin that specifically binds to the alpha chain of the interleukin 5 receptor (IL-5R) expressed on eosinophils and basophils.[A31294] It inhibits the binding of IL-5 as…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAntibodies +13
Target Protein:
Interleukin-5 receptor subunit alphaLow affinity immunoglobulin gamma Fc region receptor III-A
Waktu ParuhThe half-life of Be…
Vol. DistribusiPharmacokinetic rep…
KlirensFor a subject weigh…
Genetik -
Benserazide Approved DB12783
small molecule | CAS: 322-35-0

When levodopa is used by itself as a therapy for treating Parkinson's disease, its ubiquitous metabolism into dopamine is responsible for a resultant increase in the levels of circulating dopamine in the blood and to various extracerebral tissues. This can re…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsAromatic L-amino Acid Decarboxylase Inhibitors +6
Target Protein:
Aromatic-L-amino-acid decarboxylase
Waktu ParuhThe half-life of be…
Vol. DistribusiReadily accessible …
KlirensReadily accessible …
Genetik -
Benzamidine DB03127
small molecule | CAS: 618-39-3

Deskripsi belum tersedia.

Kategori:
AmidinesEnzyme InhibitorsProtease Inhibitors +1
Target Protein:
Serine protease 1Urokinase-type plasminogen activatorSuppressor of tumorigenicity 14 protein +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzbromarone DB12319
small molecule | CAS: 3562-84-3

Benzbromarone has been used in trials studying the basic science and treatment of Heart Failure, Hyperuricemia, Chronic Kidney Disease, Abnormal Renal Function, and Gout and Asymptomatic Hyperuricemia.

Kategori:
Antigout PreparationsAntirheumatic AgentsBenzofurans +12
Target Protein:
Anoctamin-1Solute carrier family 22 member 12Multidrug resistance-associated protein 1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzethonium Approved DB11125
small molecule | CAS: 10172-60-8

Benzethonium is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties. Its salt form, benzethonium chloride, is primarily used as a skin disinfectant at concentrations of 0.1-0.2 %, which are safe and ef…

Kategori:
AminesAnti-Infective AgentsAnti-Infective Agents, Local +7
Waktu ParuhPharmacokinetic stu…
Vol. DistribusiPharmacokinetic stu…
KlirensPharmacokinetic stu…
Genetik -
Benzgalantamine Approved DB19353
small molecule | CAS: 224169-27-1

Benzgalantamine is a prodrug of [galantamine]. Gastrointestinal adverse effects are the most frequently reported side effects in patients undergoing treatment with cholinesterase inhibitors, including galantamine, and are often a reason for treatment disconti…

Kategori:
AlkaloidsAlzheimer Disease, drug therapyAmaryllidaceae Alkaloids +11
Target Protein:
AcetylcholinesteraseCholinesteraseNeuronal acetylcholine receptor subunit alpha-7 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzhydrocodone Approved DB15465
small molecule | CAS: 1259440-61-3

Benzhydrocodone is a benzylic prodrug of hydrocodone.[L4894] It was developed in an effort to reduce parenteral bioavailability of the active metabolite as a deterrent to abuse.[A182177] Benzhydrocodone is indicated for use in the short-term management of pai…

Kategori:
Opioids
Target Protein:
Mu-type opioid receptor
Waktu ParuhThe hydrocodone met…
Vol. DistribusiThe hydrocodone met…
KlirensThe apparent cleara…
Genetik -
Benznidazole Approved DB11989
small molecule | CAS: 22994-85-0

Benznidazole was granted accelerated approval for the treatment of Chagas disease in children 2-12 years of age by the FDA on August 29, 2017.[L939] It is the first treatment made available in the United States for Chagas disease.

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntiparasitic Agents +12
Waktu ParuhThe half life of el…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Benzocaine Approved DB01086
small molecule | CAS: 94-09-7

Benzocaine is an ester local anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings.[A231219] It is commonly used for local anesthesia in many over the counter products.[L32454,L32459,L32464] Benzocaine was first u…

Kategori:
Acids, CarbocyclicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAminobenzoates +29
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzoin Approved DB14020
small molecule | CAS: 119-53-9

Benzoin is a white crystalline compound prepared by condensation of benzaldehyde in potassium cyanide, and is used in organic syntheses. This should not be confused with benzoin gum from STYRAX (see [DB11222]). Benzoin is an FDA-approved colour additive used …

Kategori:
AcetophenonesAnti-Infective Agents, LocalKetones
Target Protein:
Liver carboxylesterase 1
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Benzoin resin Approved DB11222
biotech | CAS: 9000-05-9

Benzoin resin is a balsamic resin obtained from the bark of several species of trees in the genus _Styrax_. There are two common kinds of benzoin, benzoin Siam and benzoin Sumatra, that are obtained from different species of the _Styrax_ tree. While benzoin r…

Kategori:
AngiospermsAnti-Infective Agents, LocalBiological Products +11
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Benzonatate Approved DB00868
small molecule | CAS: 104-31-4

Benzonatate is an oral antitussive drug used in the relief and suppression of cough in patients older than ten years of age.[A5790] Currently, benzonatate is the only non-narcotic antitussive available as a prescription drug.[A189519] It works to reduce the a…

Kategori:
AlkanesAminesAntitussive Agents +8
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu ParuhThe half life of be…
Vol. DistribusiThere is limited in…
KlirensThere is limited in…
Genetik -
Benzphetamine Approved DB00865
small molecule | CAS: 156-08-1

A sympathomimetic agent with properties similar to dextroamphetamine. It is used in the treatment of obesity. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1222)

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +28
Target Protein:
Synaptic vesicular amine transporterAlpha-2A adrenergic receptorAlpha-1A adrenergic receptor +1
Waktu Paruh16 to 31 hours
Vol. Distribusi-
Klirens-
Genetik -
Benzquinamide DB00767
small molecule | CAS: 63-12-7

Benzquinamide is a discontinued antiemetic compound with antihistaminic, mild anticholinergic, and sedative properties. The mechanism of action is not known, but presumably benzquinamide works via antagonism of muscarinic acetycholine receptors and histamine …

Kategori:
Agents producing tachycardiaAnticholinergic AgentsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M1 +3
Waktu Paruh1-1.6 hours (for al…
Vol. Distribusi-
Klirens-
Genetik -
Benzyl benzoate Approved DB00676
small molecule | CAS: 120-51-4

Benzyl benzoate is one of the older preparations used to treat scabies. Scabies is a skin infection caused by the mite sarcoptes scabiei. It is characterised by severe itching (particularly at night), red spots, and may lead to a secondary infection. Benzyl b…

Kategori:
AcaricidesAcids, CarbocyclicAgrochemicals +8
Target Protein:
Hormone-sensitive lipase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 451–500 dari 3253
Sebelumnya Halaman 10 / 66 Berikutnya