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Total database: 17430
Struktur (SMILES)
29 (43.3%)
Target
34 (50.7%)
Genomik
0 (0%)
Referensi
67 (100.0%)

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Hasil Pencarian (67)

Halaman 1 / 2
small molecule

Deskripsi belum tersedia.

Target Protein:
Nitric oxide synthase, inducible
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Acetylcarnitine Approved DB08842
small molecule | CAS: 3040-38-8

Acetylcarnitine is an investigational drug in the United states, Italy, United Kingdom, China, Israel, and Norway, and it is approved in Italy, Portugal, Argentina, Chile, Philippines, Australia, and India. Acetylcarnitine can be synthesized, but it is also n…

Kategori:
AminesCentral Nervous System AgentsMicronutrients +6
Waktu Paruh-
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Allysine DB02571
small molecule | CAS: 6665-12-9

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAdipatesAmino Acids +3
Target Protein:
Glutaminase-asparaginase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Anbenitamab DB18411
biotech | CAS: 2367012-88-0

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
biotech | CAS: 2636710-07-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
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AOC 1001 DB18620
biotech | CAS: 2653183-66-3

Delpacibart (AOC 1001) is being investigated in a global study for the treatment of Myotonic Dystrophy type 1 (DM1) in clinical trial NCT06411288

Waktu Paruh-
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Astodrimer DB11854
biotech | CAS: 1379746-42-5

Astodrimer has been used in trials studying the treatment and prevention of Bacterial Vaginosis. It is a lysine-based dendrimer with naphthalene disulfonic acid surface groups.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +10
Target Protein:
Envelope glycoprotein gp160
Waktu Paruh-
Vol. Distribusi-
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Barzolvolimab DB18934
biotech | CAS: 2438203-51-9

Barzolvolimab is under investigation in clinical trial NCT06455202 (A Phase 3 Study of Barzolvolimab in Participants With Chronic Spontaneous Urticaria (CSU)).

Waktu Paruh-
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Benzylpenicilloyl polylysine Approved DB00895
small molecule | CAS: 31855-75-1

Benzylpenicilloyl polylysine is used as a skin-testing reagent to detect immunoglobulin E antibodies in people with a history of penicillin allergy. The quantitation of in vitro IgE antibodies to the benzylpenicilloyl determinant is a useful tool for evaluati…

Kategori:
AcetamidesAmidesAnti-Bacterial Agents +9
Target Protein:
High affinity immunoglobulin epsilon receptor subunit gammaHigh affinity immunoglobulin epsilon receptor subunit alpha
Waktu Paruh-
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Genetik -
Cadaverine DB03854
small molecule | CAS: 462-94-2

Cadaverine is a foul-smelling diamine formed by bacterial decarboxylation of lysine.

Kategori:
AminesBiogenic AminesBiogenic Polyamines +8
Target Protein:
Carbonic anhydrase 4Carbonic anhydrase 1Carbonic anhydrase 6 +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Canoctakin DB18195
biotech | CAS: 1019859-03-0

Deskripsi belum tersedia.

Waktu Paruh-
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CTCE-9908 DB05625
small molecule | CAS: 1030384-98-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and Proteins
Target Protein:
C-X-C chemokine receptor type 4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
D-Lysine DB03252
small molecule | CAS: 923-27-3

An essential amino acid. It is often added to animal feed. [PubChem]

Target Protein:
Alanine racemase, catabolicDiaminopimelate decarboxylase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Dansyllysine DB04676
small molecule | CAS: 1101-84-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +1
Target Protein:
Immunoglobulin heavy constant alpha 2
Waktu Paruh-
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Genetik -
Dazukibart DB18429
biotech | CAS: 2639474-65-8

Deskripsi belum tersedia.

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Denecimig DB18426
biotech | CAS: 2488745-86-2

Delpacibart is a humanized, bispecific, bivalent monoclonal antibody against coagulation factor 9.

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Domvanalimab DB18848
biotech | CAS: 2368219-35-4

Domvanalimab is under investigation in clinical trial NCT05502237 (Zimberelimab and Domvanalimab in Combination With Chemotherapy Versus Pembrolizumab With Chemotherapy in Patients With Untreated Metastatic Non-small Cell Lung Cancer).

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Duvakitug DB19444
biotech | CAS: 2750005-84-4

Duvakitug is under investigation in clinical trial NCT05668013 (A Study to Evaluate the Long-term Effect of TEV-48574 in Moderate to Severe Ulcerative Colitis or Crohn's Disease).

Waktu Paruh-
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EB05 DB16477
biotech | CAS: 2641646-59-3

EB05, in combination with standard of care (SOC), is being investigated in clinical trial NCT04401475 to evaluate its safety and efficacy in adult hospitalized patients with COVID-19 and ARDS.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
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Elapegademase Approved DB14712
biotech | CAS: 1709806-75-6

Elapegademase is a PEGylated recombinant adenosine deaminase. It can be defined molecularly as a genetically modified bovine adenosine deaminase with a modification in cysteine 74 for serine and with about 13 methoxy polyethylene glycol chains bound via carbo…

Kategori:
Adenosine Deaminase InhibitorsAdjuvants, ImmunologicAmino Acids, Peptides, and Proteins +12
Target Protein:
Adenosine
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
small molecule | CAS: 1188-07-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +1
Waktu Paruh-
Vol. Distribusi-
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Evalstotug DB19410
biotech | CAS: 2460399-39-5

Evalstotug is under investigation in clinical trial NCT05271604 (A Phase 2 Open Label Study of BA3021 in Patients With Recurrent or Metastatic Squamous Cell Carcinoma of the Head and Neck).

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Exlinkibart DB17474
biotech | CAS: 2642171-64-8

Deskripsi belum tersedia.

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Felypressin DB00093
biotech | CAS: 56-59-7

A synthetic nonapeptide comprising cysteinyl, phenylalanyl, phenylalanyl, glutaminyl, asparaginyl, cysteinyl, prolyl, lysyl, and glycinamide residues in sequence, with a disulfide bridge joining the two cysteine residues. Its antidiuretic effects are less tha…

Kategori:
Amino Acids, Peptides, and ProteinsCardiovascular AgentsHormones +12
Target Protein:
Vasopressin V1a receptor
Waktu Paruh-
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Fepixnebart DB19079
biotech | CAS: 1799706-87-8

Fepixnebart is under investigation in clinical trial NCT04456686 (Chronic Pain Master Protocol (CPMP): A Study of LY3016859 in Participants With Osteoarthritis).

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Glatiramer Approved DB05259
biotech | CAS: 28704-27-0

Glatiramer acetate is a mix of synthetic polypeptides that includes L-glutamic acid, L-alanine, L-tyrosine, and L-lysine at an average molar fraction of 0.141, 0.427, 0.095, and 0.338, respectively.[L41940] Since glatiramer acetate is a heterogeneous drug, th…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +5
Target Protein:
MHC class II protein complex
Waktu ParuhNot available.
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Hiltonol DB17293
biotech | CAS: 59789-29-6

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAmino AcidsAmino Acids, Basic +17
Waktu Paruh-
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Genetik -
Insulin degludec Approved DB09564
biotech | CAS: 844439-96-9

Insulin degludec is an ultra-long-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes.[A18561,A18562,A18563,A18564,A174934] Insulin is typically prescribed for the management of diabetes mellitus to mimic the ac…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +13
Target Protein:
InsulinInsulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhThe half-life after…
Vol. DistribusiUsing a one-compart…
KlirensThe mean apparent c…
Genetik -
Insulin detemir Approved DB01307
biotech | CAS: 169148-63-4

Insulin detemir is a long-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes.[A2358, A2359, A2360, A44] Insulin is typically prescribed for the management of diabetes mellitus to mimic the activity of endogenou…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +13
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhAfter subcutaneous …
Vol. DistribusiInsulin detemir has…
KlirensThe apparent cleara…
Genetik -
Insulin glulisine Approved DB01309
biotech | CAS: 207748-29-6

Insulin glulisine is a short-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes. Insulin is typically prescribed for the management of diabetes mellitus to mimic the activity of endogenously produced human insu…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +15
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhElimination half li…
Vol. Distribusi13 L
Klirens-
Genetik -
Insulin lispro Approved DB00046
biotech | CAS: 133107-64-9

Insulin lispro is a rapid-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes. Insulin is prescribed for the management of diabetes mellitus to mimic the activity of endogenously produced human insulin, a peptid…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +14
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhAfter subcutaneous …
Vol. DistribusiWhen administered i…
KlirensWhen administered i…
Genetik -
Interferon alfa-2a Approved DB00034
biotech | CAS: 76543-88-9

Interferon a (human leukocyte protein moiety reduced). A type I interferon consisting of 165 amino acid residues with lysine in position 23. This protein is produced by recombinant DNA technology and resembles interferon secreted by leukocytes. It is used ext…

Kategori:
Adjuvants, ImmunologicAlfa InterferonsAmino Acids, Peptides, and Proteins +20
Target Protein:
Interferon alpha/beta receptor 1Interferon alpha/beta receptor 2
Waktu ParuhThe IM half-life of…
Vol. Distribusi* 0.223 to 0.748 L/…
Klirens* 2.14 - 3.62 mL/mi…
Genetik -
L-homoarginine DB03974
small molecule | CAS: 156-86-5

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +2
Target Protein:
Nitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-Saccharopine DB04207
small molecule | CAS: 997-68-2

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +1
Target Protein:
Alpha-aminoadipic semialdehyde synthase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Liraglutide Approved DB06655
biotech | CAS: 204656-20-2

Victoza contains liraglutide, a synthetic analog of human glucagon-like peptide-1(GLP-1) and acts as a GLP-1 receptor agonist.[Label,A6932] Liraglutide is 97% similar to native human GLP-1, differing primarily by substituting arginine for lysine at position 3…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +17
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhTerminal half life …
Vol. Distribusi13L[Label].
Klirens1.2L/h[Label].
Genetik -
Lisdexamfetamine Approved DB01255
small molecule | CAS: 608137-32-2

Lisdexamfetamine is a prodrug of [dextroamphetamine], a central nervous system stimulant known as d-amphetamine,[A40246] covalently attached to the naturally occurring amino acid L-lysine.[A2230] Lisdexamfetamine is the first chemically formulated prodrug sti…

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +17
Target Protein:
Trace amine-associated receptor 1
Waktu ParuhPlasma concentratio…
Vol. DistribusiDextroamphetamine, …
Klirens-
Genetik -
Lonigutamab DB18940
biotech | CAS: 2362015-67-4

Lonigutamab is under investigation in clinical trial NCT05683496 (Efficacy and Safety of Lonigutamab in Subjects With Thyroid Eye Disease (TED)).

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Lucinactant Approved DB04897
biotech | CAS: 825600-90-6

Lucinactant is a new synthetic peptide-containing surfactant for intratracheal use. It contains sinapultide, a novel, hydrophobic, 21-amino acid peptide (leucine and lysine repeating units, KL4 peptide) designed to mimic human surfactant protein-B (SB-P). Mor…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +11
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Lymecycline Approved DB00256
small molecule | CAS: 992-21-2

Lymecycline is a broad-spectrum second-generation tetracycline antibiotic used for the treatment of acne and other susceptible bacterial infections.[L13880,L13883] It has been proven a cost-effective alternative to treatment with [minocycline] with comparable…

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
30S ribosomal protein S4
Waktu ParuhThe half-life of ly…
Vol. DistribusiLymecycline is lipo…
KlirensLymecycline is part…
Genetik -
Lypressin Approved DB14642
small molecule | CAS: 50-57-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntidiuretic AgentsCardiovascular Agents +20
Target Protein:
Vasopressin V1a receptorVasopressin V2 receptorVasopressin V1b receptor
Waktu Paruh-
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Genetik -
Lysine Approved DB00123
small molecule | CAS: 56-87-1

Lysine (abbreviated as Lys or K) is an ?-amino acid with the chemical formula HO2CCH(NH2)(CH2)4NH2. This amino acid is an essential amino acid, which means that humans cannot synthesize it. Its codons are AAA and AAG. Lysine is a base, as are arginine and his…

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +10
Target Protein:
High affinity cationic amino acid transporter 1Cationic amino acid transporter 4Cationic amino acid transporter 3 +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 2Beta-lactamase OXA-10UDP-N-acetylmuramoylalanine--D-glutamate ligase +16
Waktu Paruh-
Vol. Distribusi-
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Genetik -
MALP-2 DB18482
small molecule | CAS: 250718-44-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsLipidsMacrophage Activation +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Maxy-G34 DB05718
biotech

MAXY-G34 is a pegylated variant of human granulocyte-colony stimulating factor (G-CSF). This variant contains multiple non-naturally occurring lysines that have been introduced into alpha helixes of wild type human G-CSF as PEGylation sites, and from which mu…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +15
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 2460400-64-8

Mecbotamab vedotin is an anti-Axl humanized monoclonal antibody conjugated to monomethyl auristatin E using a cleavable linker (CAB-Axl-ADC).[A255212]

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Melphalan Approved DB01042
small molecule | CAS: 148-82-3

Melphalan is a nitrogen mustard or bischloroethylamine type alkylating agent.[L40928] It was first synthesized in the early 1950s by substituting L-phenylalanine for the methyl group on nitrogen mustard.[A261150, A261155] Melphalan is used in the treatment of…

Kategori:
Alkylating ActivityAlkylating DrugsAmino Acids +17
Target Protein:
DNA
Waktu ParuhIn patients given a…
Vol. DistribusiThe volume of distr…
KlirensAverage total body …
Genetik -
small molecule | CAS: 2440-59-7

Deskripsi belum tersedia.

Target Protein:
Kynurenine--oxoglutarate transaminase 1Ornithine decarboxylaseAdenosylmethionine-8-amino-7-oxononanoate aminotransferase +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

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Genetik -
Nacystelyn DB17839
small molecule | CAS: 89344-48-9

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
4-hydroxy-tetrahydrodipicolinate synthase
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